-
analog of
lidocaine, but with reduced first-pass
metabolism.
-
used for
treatment of ventricular arrhythmias.
-
suitable
for oral administration.
-
similar
electrophysiologically to lidocaine.
-
tremor and
nausea are major dose-related adverse side
effects.
-
metabolized
by the liver.
-
Combination
with quinidine may increase efficacy and diminish
adverse effects.